SCHEMBL8712282

SCHEMBL8712282

COc1ccccc1N(CCO)S(=O)(=O)c1ccc(F)cc1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.60
KMT2A Q03164 2/20 0.49
TSHR P16473 1/20 0.49
MAPK1 P28482 1/20 0.49
HSD17B10 Q99714 1/20 0.49
KEAP1 Q14145 2/20 0.47
NFE2L2 Q16236 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HPGD P15428 2/20 0.46
LMNA P02545 1/20 0.46
POLB P06746 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8710952 0.89 ESR1 (0.60) ESR1KMT2ATSHRKEAP1NFE2L2
SCHEMBL8714947 0.89 ESR1 (0.63) ESR1KMT2ATSHRMAPK1HSD17B10
SCHEMBL10300192 0.79 ESR1 (0.49) ESR1KMT2ASMN1; SMN2HPGDLMNA
SCHEMBL18101489 0.77 SMN1; SMN2 (0.70) TSHRSMN1; SMN2HPGDLMNA
SCHEMBL9226646 0.75 HTR7 (0.59)
SCHEMBL9231944 0.74 CYP2D6 (0.54) KMT2AHSD17B10LMNA
Oxalic Acid SCHEMBL9232306 0.74 HTR7 (0.57) KMT2ATSHR
SCHEMBL9230581 0.72 HTR7 (0.66)
SCHEMBL1629150 0.72 KEAP1 (0.77) KEAP1NFE2L2
Sulfuric Acid SCHEMBL7684214 0.71 ESR1 (0.48) ESR1KMT2AHSD17B10SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed