SCHEMBL8711325

SCHEMBL8711325

CC(C)c1ccc(S(=O)(=O)NC(=O)C(Cc2ccc(Cl)cc2)c2ccc3nsnc3c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.40
ERBB2 P04626 7/20 0.40
PPARA Q07869 1/20 0.40
ITGB3 P05106 1/20 0.38
ITGAV P06756 1/20 0.38
MAPT P10636 2/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8710009 0.92 GAA (0.41) EGFRERBB2PPARAITGB3ITGAV
SCHEMBL8709894 0.92 FLT1 (0.44) EGFRERBB2PPARAITGB3ITGAV
SCHEMBL6322172 0.90 TDP1 (0.40) ITGB3ITGAVMEN1KMT2ASMN1; SMN2
SCHEMBL8712259 0.90 BMP1 (0.43) EGFRERBB2PPARAMAPTAKR1C3
SCHEMBL6320795 0.89 EDNRA (0.39) ITGB3ITGAVAKR1C3AKR1C2NPC1
SCHEMBL8712035 0.89 EDNRA (0.39) ITGB3ITGAV
SCHEMBL8709961 0.88 ITGB3 (0.36) EGFRERBB2PPARAITGB3ITGAV
SCHEMBL8708878 0.88 LARS1 (0.43) ITGB3ITGAVMAPT
SCHEMBL8709051 0.86 MAPT (0.39) EGFRERBB2PPARAITGB3ITGAV
SCHEMBL8705895 0.85 ALDH1A1 (0.41) ITGB3ITGAVMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998041515-A1 ENDOTHOLIN RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 1998-09-24 WO disclosed