SCHEMBL8711533

SCHEMBL8711533

COc1cccc(N(CCCN2CCC(C(=O)c3ccc(F)cc3)CC2)C(=O)c2ccc([N+](=O)[O-])cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.49
HTR2A P28223 3/20 0.47
ACHE P22303 1/20 0.46
MLNR O43193 1/20 0.45
DRD2 P14416 1/20 0.44
HTR2C P28335 1/20 0.44
KDM4E B2RXH2 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
HTR1A P08908 1/20 0.43
HTR1D P28221 1/20 0.43
HTR7 P34969 1/20 0.43
HTR2B P41595 1/20 0.43
CCR5 P51681 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8716772 0.95 HSD11B1 (0.51) HSD11B1HTR2AACHEMLNRDRD2
SCHEMBL8711674 0.89 HSD11B1 (0.54) HSD11B1HTR2AMLNRDRD2HTR2C
SCHEMBL8712519 0.89 HSD11B1 (0.52) HSD11B1HTR2ADRD2HTR2CKDM4E
SCHEMBL8711528 0.86 HSD11B1 (0.49) HSD11B1HTR2ACYP1A2CYP2D6ALDH1A1
SCHEMBL8716650 0.85 PTGIR (0.52) HSD11B1HTR2AACHEDRD2HTR2C
SCHEMBL9232680 0.85 HSD11B1 (0.56) HSD11B1HTR2AACHEMLNRHTR2C
Fumaric Acid SCHEMBL9234007 0.85 HSD11B1 (0.48) HSD11B1HTR2AACHEDRD2HTR2C
Fumaric Acid SCHEMBL9234015 0.85 HSD11B1 (0.48) HSD11B1HTR2AACHEDRD2HTR2C
SCHEMBL8714509 0.85 HSD11B1 (0.51) HSD11B1HTR2AACHEHTR2CKDM4E
SCHEMBL8716702 0.84 HSD11B1 (0.49) HSD11B1HTR2ADRD2HTR2CCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed