SCHEMBL8716772

SCHEMBL8716772

COc1cccc(N(CCN2CCC(C(=O)c3ccc(F)cc3)CC2)C(=O)c2ccc([N+](=O)[O-])cc2)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 5/20 0.51
HTR2A P28223 3/20 0.49
ACHE P22303 1/20 0.47
MLNR O43193 1/20 0.46
HTR2C P28335 2/20 0.46
DRD2 P14416 1/20 0.46
HTR7 P34969 2/20 0.44
HTR1A P08908 1/20 0.44
HTR1D P28221 1/20 0.44
HTR2B P41595 1/20 0.44
PTGIR P43119 1/20 0.44
HTR6 P50406 1/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8711533 0.95 HSD11B1 (0.49) HSD11B1HTR2AACHEMLNRHTR2C
SCHEMBL8711674 0.94 HSD11B1 (0.54) HSD11B1HTR2AMLNRHTR2CDRD2
SCHEMBL8716650 0.90 PTGIR (0.52) HSD11B1HTR2AACHEHTR2CDRD2
SCHEMBL9232680 0.90 HSD11B1 (0.56) HSD11B1HTR2AACHEMLNRHTR2C
SCHEMBL8714509 0.89 HSD11B1 (0.51) HSD11B1HTR2AACHEHTR2CHTR7
SCHEMBL8716656 0.88 HSD11B1 (0.54) HSD11B1HTR2AACHEHTR2CDRD2
SCHEMBL8710827 0.88 HSD11B1 (0.54) HSD11B1HTR2AACHEHTR2CDRD2
SCHEMBL8716702 0.88 HSD11B1 (0.49) HSD11B1HTR2AHTR2CDRD2HTR7
SCHEMBL8711102 0.88 HSD11B1 (0.51) HSD11B1HTR2AACHEHTR2CHTR7
Hydrochloric Acid SCHEMBL9229278 0.88 HSD11B1 (0.53) HSD11B1HTR2AACHEHTR2CDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed