SCHEMBL8712836

SCHEMBL8712836

COCOc1cc(F)c(Cl)cc1C(=O)c1ncccc1OCOC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.37
SCN9A Q15858 2/20 0.37
CLCN2 P51788 1/20 0.35
PTGES O14684 1/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
ADRA1A P35348 1/20 0.35
RAB9A P51151 4/20 0.34
NPC1 O15118 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
LMNA P02545 2/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8713191 0.95 MAPK8 (0.39) MAPK8CLCN2PTGESHTR1ADRD2
SCHEMBL8709365 0.91 GRM4 (0.37) MAPK8SCN9ACLCN2HTR1ADRD2
SCHEMBL8709890 0.90 RAB9A (0.37) MAPK8RAB9ANPC1ALDH1A1HPGD
SCHEMBL8709579 0.86 KDM4E (0.38) MAPK8RAB9AALDH1A1KMT2AMEN1
SCHEMBL8712687 0.85 POLB (0.38) CLCN2RAB9ANPC1ALDH1A1HTR2A
SCHEMBL8713114 0.84 CLCN2 (0.39) CLCN2HTR1ADRD2ADRA1AALDH1A1
SCHEMBL8710521 0.84 CNR2 (0.36) MAPK8SCN9ACLCN2RAB9AALDH1A1
SCHEMBL8715277 0.84 CLCN2 (0.38) MAPK8CLCN2RAB9AALDH1A1KMT2A
SCHEMBL8709273 0.81 XDH (0.40) CLCN2RAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL8709829 0.81 XDH (0.40) RAB9ANPC1LMNAPOLBDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed