SCHEMBL8709579

SCHEMBL8709579

COCOc1cc(F)c(Br)cc1C(=O)c1ncccc1OCOC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
APAF1 O14727 1/20 0.37
TDP2 O95551 1/20 0.37
NSD2 O96028 1/20 0.37
CASP3 P42574 1/20 0.37
PPP1CA P62136 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
SAE1 Q9UBE0 1/20 0.37
UBA2 Q9UBT2 1/20 0.37
MAPT P10636 2/20 0.35
P2RY1 P47900 1/20 0.35
RAB9A P51151 1/20 0.34
ADORA2A P29274 1/20 0.34
DHODH Q02127 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8714963 0.92 PPIA (0.43) ALDH1A1
SCHEMBL8709890 0.90 RAB9A (0.37) KDM4EALDH1A1P2RY1RAB9AADORA2A
SCHEMBL8715277 0.86 CLCN2 (0.38) KDM4EALDH1A1APAF1TDP2NSD2
SCHEMBL8712836 0.86 MAPK8 (0.37) ALDH1A1RAB9ADHODHMAPK8MEN1
SCHEMBL8713191 0.84 MAPK8 (0.39) KDM4EALDH1A1RAB9ADHODHMAPK8
SCHEMBL8024858 0.84 ALDH1A1 (0.39) KDM4EALDH1A1APAF1NSD2CASP3
SCHEMBL8710246 0.83 XDH (0.40) KDM4EALDH1A1APAF1TDP2NSD2
SCHEMBL8709054 0.82 CYP3A4 (0.47) KDM4EALDH1A1MAPTCYP3A4CYP2D6
SCHEMBL8709829 0.81 XDH (0.40) RAB9ADHODHCYP3A4CYP2C19
SCHEMBL8709365 0.80 GRM4 (0.37) KDM4EALDH1A1RAB9AMAPK8MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed