SCHEMBL8712907

SCHEMBL8712907

COCOCOC.Cc1ccc(O)c(Br)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.42
ALOX15 P16050 4/20 0.41
TDP1 Q9NUW8 3/20 0.41
TP53 P04637 2/20 0.41
ALDH1A1 P00352 3/20 0.38
HSD17B10 Q99714 2/20 0.38
L3MBTL1 Q9Y468 7/20 0.38
MAPT P10636 6/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
HPGD P15428 3/20 0.37
ALOX12 P18054 2/20 0.37
LMNA P02545 2/20 0.37
GAA P10253 1/20 0.37
AMY1A P0DUB6 1/20 0.37
KDM4E B2RXH2 2/20 0.37
USP2 O75604 1/20 0.37
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712909 0.83 TRPA1 (0.50) TRPA1ALOX15TDP1TP53ALDH1A1
SCHEMBL31501478 0.82
SCHEMBL358697 0.82
Ammonia Solution, Strong SCHEMBL28843903 0.80 TRPA1 (0.56) TRPA1ALOX15TDP1TP53ALDH1A1
SCHEMBL8709353 0.79 ALOX15 (0.38) ALOX15ESR1
Zinc Ion SCHEMBL27995538 0.78 TRPA1 (0.54) TRPA1ALOX15TDP1TP53ALDH1A1
SCHEMBL28000806 0.77 TRPA1 (0.52) TRPA1ALOX15TDP1TP53ALDH1A1
SCHEMBL7674038 0.75 ESR1 (0.41) ALOX15TDP1TP53MAPTKMT2A
SCHEMBL8709364 0.75 ALOX15 (0.37) ALOX15ESR1
Phosphoric Acid SCHEMBL28139982 0.73 TRPA1 (0.48) TRPA1ALOX15TDP1TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed