SCHEMBL8709353

SCHEMBL8709353

COCOCOC.COCOCc1ccc(O)c(Br)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.38
HDAC1 Q13547 9/20 0.38
HDAC6 Q9UBN7 8/20 0.38
HSD17B3 P37058 3/20 0.36
DBH P09172 1/20 0.36
HDAC3 O15379 2/20 0.36
HDAC2 Q92769 2/20 0.36
HDAC4 P56524 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
PTPN1 P18031 1/20 0.35
CCR6 P51684 1/20 0.35
HKDC1 Q2TB90 1/20 0.35
SNCA P37840 1/20 0.34
ESR1 P03372 1/20 0.34
NCOR2 Q9Y618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8709364 0.95 ALOX15 (0.37) ALOX15HDAC1HDAC6HSD17B3DBH
SCHEMBL10907421 0.84 ALOX15 (0.45) ALOX15HDAC1HDAC6HSD17B3DBH
SCHEMBL8712907 0.79 TRPA1 (0.42) ALOX15ESR1
SCHEMBL15335397 0.79 PTPN1 (0.31) PTPN1
SCHEMBL14762230 0.77 ALOX15 (0.40) ALOX15HDAC1HDAC6HSD17B3DBH
SCHEMBL8709359 0.77 MAPT (0.38)
SCHEMBL8715513 0.76 CDK1 (0.51)
SCHEMBL500206 0.76 FFAR4 (0.32) PTPN1
SCHEMBL2960316 0.76 ALDH1A1 (0.40) PTPN1
SCHEMBL10908075 0.75 CYP3A4 (0.51) HDAC1HDAC6HDAC3HDAC2ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed