SCHEMBL8712933

SCHEMBL8712933

O=C1c2cccc3ncc(n23)CN1CCC1CCN(S(=O)(=O)C(F)(F)F)CC1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.35
HTR2A P28223 13/20 0.34
HTR1A P08908 12/20 0.34
DRD2 P14416 12/20 0.34
HTR7 P34969 12/20 0.34
HTR6 P50406 12/20 0.34
PIM1 P11309 1/20 0.33
FLT3 P36888 1/20 0.33
KCNH2 Q12809 1/20 0.33
PIM3 Q86V86 1/20 0.33
PIM2 Q9P1W9 1/20 0.33
CNR2 P34972 2/20 0.32
HTR2C P28335 1/20 0.32
CNR1 P21554 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7863415 0.93 HTR2A (0.35) ACHEHTR2AHTR1ADRD2HTR7
SCHEMBL7870234 0.88 HDAC3 (0.32) HTR2AHTR1ADRD2HTR7HTR6
Hydrochloric Acid SCHEMBL7871669 0.87 HDAC3 (0.32) HTR2AHTR1ADRD2HTR7HTR6
SCHEMBL7868936 0.85 KCNH2 (0.33) PIM1FLT3KCNH2PIM3PIM2
Hydrochloric Acid SCHEMBL7863474 0.84 KCNH2 (0.32) PIM1FLT3KCNH2PIM3PIM2
SCHEMBL8589168 0.82 HTR7 (0.36) HTR2AHTR1ADRD2HTR7HTR6
Hydrochloric Acid SCHEMBL8716045 0.81 HTR7 (0.35) HTR2AHTR1ADRD2HTR7HTR6
SCHEMBL8713773 0.81 ACHE (0.34) ACHEHTR2AHTR1ADRD2HTR7
SCHEMBL8708955 0.79 HTR2A (0.35) ACHEHTR2AHTR1ADRD2HTR7
SCHEMBL8713347 0.75 HTR1A (0.34) HTR2AHTR1ADRD2HTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0826686-A2 Tricyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-03-04 EP disclosed