SCHEMBL8713352

SCHEMBL8713352

COc1cccc(N(CCN2CCC(C(=O)c3ccc(F)cc3)CC2)C(=O)c2ccccc2N)c1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 6/20 0.52
LMNA P02545 3/20 0.46
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
HTT P42858 1/20 0.45
HTR2A P28223 4/20 0.44
HTR2C P28335 2/20 0.44
DRD2 P14416 1/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C19 P33261 1/20 0.44
GRM2 Q14416 1/20 0.44
HTR7 P34969 1/20 0.44
HTR6 P50406 1/20 0.44
KDM4E B2RXH2 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8710827 0.89 HSD11B1 (0.54) HSD11B1LMNAALDH1A1SMN1; SMN2HTT
Hydrochloric Acid SCHEMBL9229278 0.88 HSD11B1 (0.53) HSD11B1LMNAKMT2AALDH1A1SMN1; SMN2
SCHEMBL8714991 0.88 HSD11B1 (0.51) HSD11B1LMNAKMT2AALDH1A1SMN1; SMN2
SCHEMBL8713835 0.88 HSD11B1 (0.51) HSD11B1LMNAKMT2AALDH1A1SMN1; SMN2
SCHEMBL8716461 0.88 HSD11B1 (0.55) HSD11B1LMNAALDH1A1SMN1; SMN2HTT
SCHEMBL8712025 0.87 CYP2D6 (0.49) HSD11B1LMNAKMT2AALDH1A1SMN1; SMN2
SCHEMBL8716702 0.87 HSD11B1 (0.49) HSD11B1LMNAKMT2AALDH1A1SMN1; SMN2
SCHEMBL8716656 0.86 HSD11B1 (0.54) HSD11B1LMNAALDH1A1SMN1; SMN2HTT
SCHEMBL8711204 0.85 HSD11B1 (0.48) HSD11B1LMNAKMT2ASMN1; SMN2HTT
Hydrochloric Acid SCHEMBL8711167 0.85 HSD11B1 (0.53) HSD11B1LMNAALDH1A1SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed