SCHEMBL8713835

SCHEMBL8713835

COc1cccc(N(CCN2CCC(C(=O)c3ccc(F)cc3)CC2)C(=O)c2ccc(N)c(C)c2)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.51
HTR2A P28223 3/20 0.44
HTR2C P28335 3/20 0.44
DRD2 P14416 1/20 0.44
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTR7 P34969 2/20 0.43
HTR6 P50406 2/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HTT P42858 1/20 0.43
TNKS O95271 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
KMT2A Q03164 1/20 0.42
PTGIR P43119 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8714991 0.92 HSD11B1 (0.51) HSD11B1HTR2AHTR2CDRD2CYP2D6
SCHEMBL8714653 0.91 OPRM1 (0.51) HSD11B1HTR2AHTR2CDRD2CYP2C19
SCHEMBL8716461 0.90 HSD11B1 (0.55) HSD11B1HTR2AHTR2CDRD2HTR7
SCHEMBL8710827 0.90 HSD11B1 (0.54) HSD11B1HTR2AHTR2CDRD2HTR7
Hydrochloric Acid SCHEMBL9229278 0.89 HSD11B1 (0.53) HSD11B1HTR2AHTR2CDRD2HTR7
SCHEMBL8713352 0.88 HSD11B1 (0.52) HSD11B1HTR2AHTR2CDRD2CYP2D6
SCHEMBL8715758 0.88 HSD11B1 (0.48) HSD11B1HTR2AHTR2CDRD2CYP2D6
SCHEMBL8716656 0.87 HSD11B1 (0.54) HSD11B1HTR2AHTR2CDRD2HTR7
Fumaric Acid SCHEMBL9231642 0.86 HSD11B1 (0.50) HSD11B1HTR2AHTR2CDRD2CYP2D6
Fumaric Acid SCHEMBL9231639 0.86 HSD11B1 (0.50) HSD11B1HTR2AHTR2CDRD2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed