SCHEMBL8713424

SCHEMBL8713424

N#Cc1ccc2oc(C(=O)Cl)cc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.48
CYP2A6 P11509 1/20 0.45
PLAU P00749 1/20 0.44
FLT3 P36888 3/20 0.44
GPR35 Q9HC97 1/20 0.42
MAOB P27338 1/20 0.42
ALDH1A1 P00352 2/20 0.41
PIM1 P11309 2/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
CASP1 P29466 1/20 0.41
BRCA1 P38398 1/20 0.41
CASP7 P55210 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PGR P06401 2/20 0.41
NOS3 P29474 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1819421 0.85 PIM1 (0.58) HRH3CYP2A6PLAUFLT3ALDH1A1
SCHEMBL7384075 0.84 ALDH1A1 (0.61) HRH3CYP2A6PLAUFLT3MAOB
SCHEMBL9231951 0.80 CA12 (0.46) HRH3CYP2A6PLAUFLT3ALDH1A1
SCHEMBL7384685 0.80 GSK3B (0.49) HRH3CYP2A6PLAUFLT3ALDH1A1
SCHEMBL7389709 0.78 DRD2 (0.44) HRH3CYP2A6PLAUFLT3ALDH1A1
SCHEMBL7449870 0.77 CA12 (0.50) HRH3MAOBALDH1A1KDM4EHPGD
SCHEMBL3613922 0.76 MAOB (0.63) FLT3GPR35MAOBALDH1A1KDM4E
SCHEMBL9989803 0.76 FLT3 (0.73) FLT3MAOBALDH1A1PIM1KDM4E
SCHEMBL23875930 0.75 NPC1 (0.47) PLAUFLT3MAOBALDH1A1PIM1
SCHEMBL3619989 0.75 PIM1 (0.72) CYP2A6FLT3GPR35ALDH1A1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011159781-A2 BITTER TASTE MODULATORS SENOMYX, INC. (US) 2011-12-22 WO disclosed
US-5753670-A ANTICOAGULANTS THE GREEN CROSS CORPORATION (JP) 1998-05-19 US disclosed
US-5635527-A ANTAGONIST OF PLATELET MEMBRANE GLYCOPROTEIN; TREATMENT OF THROMBOTIC DISEASES THE GREEN CROSS CORPORATION (JP) 1997-06-03 US disclosed
EP-0712844-A1 NOVEL FUSED-RING CARBOXYLIC ACID COMPOUND OR SALT THEREOF, AND MEDICINAL USE THEREOF THE GREEN CROSS CORPORATION (JP) 1996-05-22 EP disclosed