SCHEMBL8714137

SCHEMBL8714137

CC(C)c1ccc(S(=O)(=O)NC(=O)C(Cc2cccc(Oc3ccccc3)c2)c2ccc3nsnc3c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TARS1 P26639 1/20 0.45
FFAR1 O14842 3/20 0.40
ITGB3 P05106 1/20 0.40
ITGAV P06756 1/20 0.40
CTSK P43235 2/20 0.39
CTSS P25774 1/20 0.39
MME P08473 1/20 0.39
ACE P12821 1/20 0.39
CPA1 P15085 1/20 0.39
ACE2 Q9BYF1 1/20 0.39
FDFT1 P37268 2/20 0.37
BCL2L1 Q07817 2/20 0.37
MCL1 Q07820 2/20 0.37
MMP9 P14780 2/20 0.37
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37
MMP3 P08254 1/20 0.37
MMP7 P09237 1/20 0.37
MMP13 P45452 1/20 0.37
PTGES O14684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8706028 0.92 MAPT (0.41) TARS1FFAR1ITGB3ITGAVCTSK
SCHEMBL8706016 0.91 NPC1 (0.44) ITGB3ITGAVMMP13MAPT
SCHEMBL8709540 0.89 ITGB3 (0.43) ITGB3ITGAVCTSKCTSSMMP9
SCHEMBL8709039 0.88 BCL9 (0.40) ITGB3ITGAVMMP9MMP2MMP13
SCHEMBL8711199 0.87 MRGPRX4 (0.41) ITGB3ITGAVMMP13MAPT
SCHEMBL8708878 0.87 LARS1 (0.43) TARS1ITGB3ITGAVMMEACE
SCHEMBL8705444 0.86 PTGES (0.43) ITGB3ITGAVPTGESMAPT
SCHEMBL8705895 0.86 ALDH1A1 (0.41) TARS1ITGB3ITGAVMAPT
SCHEMBL8707231 0.85 SLC7A5 (0.39) ITGB3ITGAVMMP13MAPT
SCHEMBL8709051 0.85 MAPT (0.39) ITGB3ITGAVMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998041515-A1 ENDOTHOLIN RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 1998-09-24 WO disclosed