SCHEMBL8714653

SCHEMBL8714653

COc1ccc(N(CCN2CCC(C(=O)c3ccc(F)cc3)CC2)C(=O)c2ccc(N)c(C)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.51
PTGIR P43119 1/20 0.49
ALDH1A1 P00352 2/20 0.49
LMNA P02545 2/20 0.49
HSD11B1 P28845 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
KMT2A Q03164 1/20 0.47
SLC18A3 Q16572 4/20 0.46
DRD2 P14416 2/20 0.46
CYP1A2 P05177 1/20 0.46
GAA P10253 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HTR2A P28223 2/20 0.46
HTR2C P28335 2/20 0.46
POLB P06746 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
HTR7 P34969 1/20 0.45
HTR6 P50406 1/20 0.45
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712582 0.92 OPRM1 (0.51) OPRM1PTGIRALDH1A1LMNAHSD11B1
SCHEMBL8713835 0.91 HSD11B1 (0.51) PTGIRALDH1A1LMNAHSD11B1SMN1; SMN2
SCHEMBL8711336 0.89 PTGIR (0.55) OPRM1PTGIRALDH1A1LMNAHSD11B1
SCHEMBL8716576 0.87 OPRM1 (0.48) OPRM1PTGIRALDH1A1LMNAHSD11B1
SCHEMBL8713866 0.87 OPRM1 (0.48) OPRM1PTGIRALDH1A1LMNAHSD11B1
SCHEMBL8711220 0.86 PTGIR (0.56) OPRM1PTGIRALDH1A1LMNAHSD11B1
SCHEMBL8716637 0.85 PTGIR (0.54) OPRM1PTGIRALDH1A1LMNAHSD11B1
Fumaric Acid SCHEMBL9230497 0.84 PTGIR (0.53) OPRM1PTGIRALDH1A1LMNAHSD11B1
Fumaric Acid SCHEMBL9230503 0.84 PTGIR (0.53) OPRM1PTGIRALDH1A1LMNAHSD11B1
SCHEMBL8716650 0.84 PTGIR (0.52) OPRM1PTGIRALDH1A1LMNAHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed