SCHEMBL8714915

SCHEMBL8714915

Oc1[c]cc(Nc2ccc(F)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.39
KMT2A Q03164 5/20 0.39
POLB P06746 1/20 0.39
DHODH Q02127 2/20 0.38
GAA P10253 1/20 0.37
ALDH1A1 P00352 3/20 0.35
MAPT P10636 3/20 0.34
MAPK10 P53779 1/20 0.34
ALOX5 P09917 2/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
ALOX12 P18054 2/20 0.33
TXN P10599 1/20 0.33
PRKD3 O94806 1/20 0.33
EGFR P00533 1/20 0.33
PRKCG P05129 1/20 0.33
PRKCB P05771 1/20 0.33
SRC P12931 1/20 0.33
PRKCA P17252 1/20 0.33
PRKCH P24723 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL303555 0.75
SCHEMBL395770 0.75 ALDH1A1 (0.50) MEN1KMT2APOLBGAAALDH1A1
SCHEMBL1028204 0.73 GAA (0.61) MEN1KMT2APOLBDHODHGAA
SCHEMBL8715505 0.68 MEN1 (0.42) MEN1KMT2APOLBDHODHALDH1A1
SCHEMBL21560850 0.68 TXN (0.57) MEN1KMT2APOLBALDH1A1MAPT
SCHEMBL4579384 0.68 TXN (0.57) MEN1KMT2APOLBALDH1A1MAPT
Cyclooctane SCHEMBL8134205 0.68 KMT2A (0.45) MEN1KMT2APOLBALDH1A1MAPT
SCHEMBL3932395 0.67 MEN1 (0.40) MEN1KMT2APOLBDHODHALDH1A1
SCHEMBL904596 0.66 ALDH1A1 (0.72) MEN1KMT2APOLBALDH1A1MAPT
SCHEMBL25354895 0.64 MEN1 (0.59) MEN1KMT2APOLBALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763596-A PYROLO PYRIMIDINE AND PYRAZOLO PYRIMIDINE COMPOUMDS; TREATMENT OF CARDIOVASCULAR AND BRAIN DISORDERS, ANTIINFLAMMATORY AGENTS METABASIS THERAPEUTICS, INC. (US) 1998-06-09 US disclosed
US-5674998-A FOR TREATING CARDIOVASCULAR OR BRAIN DISORDERS, OR AS ANTIINFLAMMATORY AGENT GENSIA INC. (US) 1997-10-07 US disclosed