SCHEMBL8715515

SCHEMBL8715515

COCOCc1ccc(O)c(C=O)c1.COOC

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.50
ERN1 O75460 14/20 0.47
TRIM24 O15164 1/20 0.41
TYR P14679 1/20 0.41
TRIM33 Q9UPN9 1/20 0.41
NT5E P21589 1/20 0.39
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8715513 0.95 CDK1 (0.51) CDK1ERN1TRIM24TYRTRIM33
SCHEMBL17967100 0.84 CDK1 (0.59) CDK1ERN1TRIM24TYRTRIM33
SCHEMBL8709364 0.77 ALOX15 (0.37)
SCHEMBL2963284 0.77 ERN1 (0.37) ERN1TRIM24TYRTRIM33LMNA
SCHEMBL11518506 0.75 CDK1 (0.51) CDK1ERN1TRIM24TYRTRIM33
SCHEMBL2980854 0.73 ERN1 (0.33) CDK1ERN1LMNAMAPT
SCHEMBL15543635 0.73 CDK1 (0.71) CDK1ERN1TRIM24TYRTRIM33
SCHEMBL21137127 0.72 KDM4E (0.47) CDK1ERN1LMNAMAPT
SCHEMBL305074 0.72 CDK1 (0.65) CDK1ERN1TRIM24TRIM33NT5E
SCHEMBL8709353 0.72 ALOX15 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed