SCHEMBL8716657

SCHEMBL8716657

Cc1c(Cl)cccc1N1C(=O)CN(c2ccccc2)C1=S

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 11/20 0.51
MEN1 O00255 10/20 0.51
GAA P10253 2/20 0.46
ALOX15 P16050 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
RECQL P46063 1/20 0.45
HCRTR1 O43613 1/20 0.41
P2RX7 Q99572 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8710997 0.82 MEN1 (0.54) KMT2AMEN1GAAALOX15RECQL
SCHEMBL1685398 0.79 KMT2A (0.56) KMT2AMEN1GAANPC1RAB9A
SCHEMBL8711085 0.77 KMT2A (0.51) KMT2AMEN1GAANPC1RAB9A
SCHEMBL11072116 0.77 KMT2A (0.49) KMT2AMEN1GAANPC1RAB9A
SCHEMBL11065342 0.77 HTT (0.53) KMT2AMEN1GAANPC1RAB9A
SCHEMBL11067046 0.76 KMT2A (0.56) KMT2AMEN1GAANPC1RAB9A
SCHEMBL8661222 0.73 MEN1 (0.48) KMT2AMEN1GAAALOX15RECQL
SCHEMBL11563108 0.70 HPGD (0.54) KMT2AMEN1GAAALOX15RECQL
SCHEMBL5955047 0.69 KMT2A (0.56) KMT2AMEN1GAANPC1RAB9A
SCHEMBL5955275 0.69 KMT2A (0.56) KMT2AMEN1GAANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821372-A USEFUL FOR INCREASING BLOOD SERUM HIGH DENSITY LIPOPROTEIN LEVELS(HDL) AMERICAN HOME PRODUCTS CORPORATION (US) 1998-10-13 US claimed
US-5821372-A USEFUL FOR INCREASING BLOOD SERUM HIGH DENSITY LIPOPROTEIN LEVELS(HDL) AMERICAN HOME PRODUCTS CORPORATION (US) 1998-10-13 US disclosed
US-5554607-A INCREASING HDL CHOLESTEROL AMERICAN HOME PRODUCTS CORPORATION (US) 1996-09-10 US disclosed