SCHEMBL8716890

SCHEMBL8716890

O=[C]OC(C(=O)OCc1ccccc1)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.47
NPC1 O15118 1/20 0.47
ITGA4 P13612 1/20 0.46
ITGB7 P26010 1/20 0.46
PPIA P62937 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
IDO1 P14902 1/20 0.42
MAPT P10636 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42
ATM Q13315 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5481199 0.95 RAB9A (0.49) RAB9ANPC1ITGA4ITGB7TDP1
SCHEMBL7294874 0.88 IDO1 (0.43) RAB9AIDO1MAPTALDH1A1HTT
SCHEMBL10569475 0.88 MAPT (0.45) RAB9ANPC1IDO1MAPTALDH1A1
SCHEMBL3861174 0.88 IDO1 (0.43) RAB9AIDO1MAPTALDH1A1HTT
SCHEMBL4438089 0.86 GAA (0.53) RAB9AMAPTALDH1A1HTTATM
SCHEMBL7278760 0.86 GAA (0.53) RAB9AMAPTALDH1A1HTTATM
SCHEMBL212215 0.85 ALDH1A1 (0.51) TDP1ALDH1A1NPSR1
SCHEMBL11004392 0.83 ALOX5 (0.56) RAB9ATDP1MAPTALDH1A1HTT
SCHEMBL9368647 0.82 RAB9A (0.46) RAB9ANPC1IDO1ALDH1A1
SCHEMBL9050930 0.82 MEN1 (0.43) RAB9AIDO1MAPTALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5834486-A ANTIPROLIFERATIVE, ANTIPROTOZOA AGENTS NOVARTIS AG (CH) 1998-11-10 US disclosed
US-5149802-A Chemical intermediates for antibiotics MERCIAN CORPORATION (JP) 1992-09-22 US disclosed
US-5096899-A Nonhydrolyzing oxapenicillins BAYER AKTIENGESELLSCHAFT (DE) 1992-03-17 US disclosed
EP-0163433-B1 ANTIBACTERIAL SOLID COMPOSITION FOR ORAL ADMINISTATION Takeda Chemical Industries, Ltd. (JP) 1990-08-01 EP disclosed
EP-0008888-B1 BETA-LACTAM ANTIBACTERIAL COMPOUNDS, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1983-09-21 EP disclosed
EP-0008888-A1 Beta-lactam antibacterial compounds, their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1980-03-19 EP disclosed