SCHEMBL8716968

SCHEMBL8716968

COc1cccc(C2C(C(C)C(C)C(N)=O)C2(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 2/20 0.48
CACNA1F O60840 1/20 0.43
CACNA1D Q01668 1/20 0.43
CACNA1S Q13698 1/20 0.43
CACNA1C Q13936 1/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
GLA P06280 2/20 0.43
GAA P10253 2/20 0.43
HPGD P15428 2/20 0.43
TSHR P16473 2/20 0.43
MAPK1 P28482 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
HSD17B10 Q99714 1/20 0.43
PARP1 P09874 1/20 0.40
KDM1A O60341 2/20 0.40
TRPM8 Q7Z2W7 2/20 0.38
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8332241 0.75 ALOX5 (0.55) SLC9A1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL8334052 0.71 SLC9A1 (0.43) SLC9A1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL8333226 0.70 SLC9A1 (0.47) SLC9A1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL8098209 0.69 MTNR1A (0.43) SLC9A1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL8098211 0.69 MTNR1A (0.43) SLC9A1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL8331760 0.68 HTR2C (0.44) SLC9A1KDM4EALDH1A1GLAGAA
SCHEMBL8332475 0.68 HTR2C (0.58) SLC9A1KDM4EALDH1A1GAAKDM1A
SCHEMBL3287384 0.68 SLC9A1 (0.56) SLC9A1KDM4EALDH1A1GLAGAA
SCHEMBL3287396 0.68 SLC9A1 (0.56) SLC9A1KDM4EALDH1A1GLAGAA
SCHEMBL3287387 0.68 SLC9A1 (0.56) SLC9A1KDM4EALDH1A1GLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed