SCHEMBL8718280

SCHEMBL8718280

COc1ccc([N+](=O)[O-])cc1CN1CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 1/20 0.61
ALDH1A1 P00352 11/20 0.57
KDM4E B2RXH2 4/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
HTT P42858 1/20 0.57
TACR1 P25103 1/20 0.57
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
HPGD P15428 2/20 0.49
TDP1 Q9NUW8 1/20 0.49
PKM P14618 1/20 0.49
USP2 O75604 1/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48
THRB P10828 1/20 0.48
CYP2D6 P10635 2/20 0.47
CTSB P07858 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7563807 0.85 ALDH1A1 (0.61) KCNJ1ALDH1A1KDM4ESMN1; SMN2HTT
Hydrochloric Acid SCHEMBL7564284 0.84 KCNJ1 (0.58) KCNJ1ALDH1A1KDM4ESMN1; SMN2HTT
SCHEMBL21044045 0.83 CTSB (0.68) ALDH1A1KDM4ESMN1; SMN2HTTMEN1
SCHEMBL8714933 0.83 CTSB (0.68) ALDH1A1KDM4ESMN1; SMN2HTTMEN1
SCHEMBL7422612 0.82 TACR1 (0.58) KCNJ1ALDH1A1KDM4ESMN1; SMN2HTT
SCHEMBL922716 0.81 KCNJ1 (0.74) KCNJ1ALDH1A1KDM4ESMN1; SMN2HTT
SCHEMBL8715361 0.81 KCNJ1 (0.55) KCNJ1ALDH1A1KDM4ESMN1; SMN2HTT
SCHEMBL6548611 0.80 TACR1 (0.53) ALDH1A1KDM4ETACR1MEN1KMT2A
SCHEMBL20272178 0.79 MAPT (0.60) KCNJ1ALDH1A1KDM4ESMN1; SMN2HTT
SCHEMBL8658728 0.79 ALDH1A1 (0.48) KCNJ1ALDH1A1KDM4ESMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0353450-B1 Macrocyclic bifunctional chelants, complexes thereof and their antibody conjugates DOW CHEMICAL CO (US) 1995-03-29 EP claimed
US-5756065-A DIAGNOSTIC CHELATES FOR ANTIBODIES AND RADIOACTIVE MATERIALS THE DOW CHEMICAL COMPANY (US) 1998-05-26 US disclosed
US-5652361-A ANTITUMOR THE DOW CHEMICAL COMPANY (US) 1997-07-29 US disclosed
US-5435990-A Chelate-antibody complexes, treatment and diagnosis of cancer, tetraazacyclododecane compounds THE DOW CHEMICAL COMPANY (US) 1995-07-25 US disclosed
EP-0353450-B1 Macrocyclic bifunctional chelants, complexes thereof and their antibody conjugates DOW CHEMICAL CO (US) 1995-03-29 EP disclosed
EP-0420942-A1 MACROCYCLIC BIFUNCTIONAL CHELANTS, COMPLEXES THEREOF AND THEIR ANTIBODY CONJUGATES THE DOW CHEMICAL COMPANY (US) 1991-04-10 EP disclosed
EP-0353450-A1 Macrocyclic bifunctional chelants, complexes thereof and their antibody conjugates THE DOW CHEMICAL COMPANY (US) 1990-02-07 EP disclosed
WO-1989012631-A1 MACROCYCLIC BIFUNCTIONAL CHELANTS, COMPLEXES THEREOF AND THEIR ANTIBODY CONJUGATES THE DOW CHEMICAL COMPANY (US) 1989-12-28 WO disclosed