SCHEMBL8720323

SCHEMBL8720323

Cc1ccc([C@H](C)C(N)N2CCCC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.42
SLC6A3 Q01959 6/20 0.40
SLC6A2 P23975 5/20 0.40
SLC6A4 P31645 3/20 0.40
TSHR P16473 2/20 0.39
ALDH1A1 P00352 2/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ADRB2 P07550 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
OPRL1 P41146 1/20 0.36
TP53 P04637 1/20 0.35
USP2 O75604 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8716792 0.84 ADRB2 (0.48) HRH3SLC6A3SLC6A2SLC6A4TSHR
SCHEMBL8717059 0.83 CYP2D6 (0.53) SLC6A3TSHRALDH1A1CHRM2CHRM1
SCHEMBL23733409 0.77 HRH3 (0.41) HRH3SLC6A3SLC6A2SLC6A4TSHR
SCHEMBL16270668 0.76 CHRM2 (0.54) HRH3SLC6A3SLC6A2SLC6A4TSHR
SCHEMBL2735673 0.76 CHRM2 (0.54) HRH3SLC6A3SLC6A2SLC6A4TSHR
SCHEMBL9491375 0.76 SLC6A3 (0.50) SLC6A3SLC6A2SLC6A4ALDH1A1SMN1; SMN2
SCHEMBL8717426 0.76 DPP4 (0.40) TSHRSMN1; SMN2OPRM1OPRD1OPRK1
SCHEMBL2491857 0.74 OPRM1 (0.51) HRH3SLC6A3SLC6A2SLC6A4TSHR
SCHEMBL31046804 0.72 CYP2D6 (0.54) HRH3SLC6A3SLC6A2SLC6A4TSHR
SCHEMBL13699289 0.71 CHRNA7 (0.42) ALDH1A1TDP1ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0569802-B1 Arylacetamides MERCK PATENT GMBH (DE) 1998-07-15 EP disclosed
EP-0569802-A1 Arylacetamides MERCK PATENT GmbH (DE) 1993-11-18 EP disclosed