SCHEMBL8716792

SCHEMBL8716792

C[C@@H](c1ccc(Cl)cc1)C(N)N1CCCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.48
SLC6A3 Q01959 5/20 0.42
SLC6A4 P31645 4/20 0.42
CYP2D6 P10635 3/20 0.42
CHRM2 P08172 3/20 0.42
CHRM1 P11229 3/20 0.42
SLC6A2 P23975 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HTR1A P08908 2/20 0.42
ADRA2A P08913 2/20 0.42
DRD1 P21728 2/20 0.42
TBXA2R P21731 2/20 0.42
ADRA1A P35348 2/20 0.42
DRD3 P35462 2/20 0.42
KCNH2 Q12809 2/20 0.42
ALDH1A1 P00352 2/20 0.42
OPRM1 P35372 1/20 0.42
USP2 O75604 1/20 0.42
CYP3A4 P08684 1/20 0.42
LMNA P02545 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8720323 0.84 HRH3 (0.42) ADRB2SLC6A3SLC6A4CYP2D6CHRM2
SCHEMBL8717059 0.81 CYP2D6 (0.53) SLC6A3CYP2D6CHRM2CHRM1ADRA2A
SCHEMBL9491375 0.81 SLC6A3 (0.50) SLC6A3SLC6A4SLC6A2SMN1; SMN2ALDH1A1
SCHEMBL8719795 0.77 DPP7 (0.43) ADRB2OPRM1DPP7DPP4
SCHEMBL22206739 0.76 CHRM2 (0.57) ADRB2SLC6A3SLC6A4CYP2D6CHRM2
SCHEMBL22206767 0.76 CHRM2 (0.57) ADRB2SLC6A3SLC6A4CYP2D6CHRM2
SCHEMBL16757326 0.71 CYP2D6 (0.66) SLC6A3SLC6A4CYP2D6CHRM2CHRM1
SCHEMBL11949354 0.71 ADRB2 (0.62) ADRB2SLC6A3SLC6A4SLC6A2LMNA
SCHEMBL6789003 0.70 TP53 (0.48) SLC6A3SLC6A4CYP2D6CHRM2CHRM1
SCHEMBL16461973 0.69 RPS6KB1 (0.50) CYP2D6CYP3A4LMNAKMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0569802-B1 Arylacetamides MERCK PATENT GMBH (DE) 1998-07-15 EP disclosed
EP-0569802-A1 Arylacetamides MERCK PATENT GmbH (DE) 1993-11-18 EP disclosed