SCHEMBL872044

SCHEMBL872044

CN(Cc1ccccc1)c1ccccc1C(=O)N1CCC[C@H]1C(=O)Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
TACR1 P25103 1/20 0.40
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
KHK P50053 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
PFKFB2 O60825 1/20 0.39
PFKFB1 P16118 1/20 0.39
PFKFB3 Q16875 1/20 0.39
PABPC1 P11940 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
KDM1A O60341 1/20 0.38
RCOR1 Q9UKL0 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845339 0.92 ALDH1A1 (0.49) ALDH1A1KDM4ELMNATACR1CYP2C9
SCHEMBL871691 0.85 ALDH1A1 (0.44) ALDH1A1KDM4ELMNACYP2C9CYP2C19
SCHEMBL10119320 0.84 ALDH1A1 (0.43) ALDH1A1KDM4ELMNACYP2C9CYP2C19
SCHEMBL874311 0.83 ALDH1A1 (0.47) ALDH1A1KDM4ELMNACYP2C9CYP2C19
SCHEMBL873465 0.83 KDM4E (0.47) ALDH1A1KDM4ELMNAPFKFB2PFKFB1
SCHEMBL10119502 0.82 CYP2C9 (0.39) ALDH1A1CYP2C9CYP2C19KHKPFKFB2
SCHEMBL874324 0.82 MAPK1 (0.42) ALDH1A1LMNACYP2C9CYP2C19PABPC1
SCHEMBL874056 0.82 TRPV1 (0.42) ALDH1A1CYP2C9CYP2C19MEN1KMT2A
SCHEMBL874313 0.81 MAPK1 (0.50) ALDH1A1LMNACYP2C9CYP2C19MEN1
SCHEMBL845110 0.81 ALDH1A1 (0.48) ALDH1A1KDM4ELMNACYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed