SCHEMBL8720565

SCHEMBL8720565

CCOC(=O)c1nccnc1Oc1ccccc1C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.51
P2RY1 P47900 5/20 0.48
SLC5A1 P13866 1/20 0.43
SLC5A2 P31639 1/20 0.43
BRD4 O60885 1/20 0.42
HTR1A P08908 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
ALDH1A1 P00352 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
NPC1 O15118 1/20 0.42
NFE2L2 Q16236 1/20 0.41
MRGPRX1 Q96LB2 1/20 0.41
CACNA1C Q13936 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8341105 0.86 P2RY1 (0.50) P2RY1HTR1ASLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL8725899 0.82 P2RY1 (0.48) P2RY1HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL18137682 0.80 BRD4 (0.56) MAPTSLC5A1SLC5A2BRD4ALDH1A1
SCHEMBL14988166 0.74 MAPK1 (0.45) MAPTP2RY1ALDH1A1NPSR1MRGPRX1
SCHEMBL25227115 0.73 MAPT (0.51) MAPTSLC5A1SLC5A2BRD4ALDH1A1
SCHEMBL28244005 0.73 BRD4 (0.55) MAPTP2RY1BRD4ALDH1A1NPSR1
SCHEMBL8723588 0.73 NPSR1 (0.46) P2RY1HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL11732040 0.73 MAPT (0.49) MAPTBRD4ALDH1A1NPSR1NPC1
SCHEMBL9852615 0.72 TRPM8 (0.59) MAPTP2RY1
SCHEMBL19924873 0.72 MAPT (0.56) MAPTBRD4ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700391-B1 HERBICIDAL COMPOUNDS SHELL INT RESEARCH (NL) 1998-10-21 EP disclosed
US-5759956-A PYRAZINE CARBOXAMIDE DERIVATIVES AMERICAN CYANAMID COMPANY (US) 1998-06-02 US disclosed
EP-0700391-A1 HERBICIDAL COMPOUNDS SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1996-03-13 EP disclosed
WO-1994027974-A1 HERBICIDAL COMPOUNDS SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ B.V. (NL) 1994-12-08 WO disclosed