SCHEMBL8720600

SCHEMBL8720600

CCCOC1(c2ccccc2)COCC2(CC(c3ccc(F)cc3)CO2)C1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.37
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8717928 0.86 TACR1 (0.40) TACR1
SCHEMBL8201358 0.77 OPRM1 (0.34) TACR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL8720765 0.76 TACR1 (0.36) TACR1
SCHEMBL8912656 0.65 TACR1 (0.46) TACR1
SCHEMBL13059859 0.62 LIG1 (0.38) TACR1
Hydrochloric Acid SCHEMBL8911488 0.62 TACR1 (0.42) TACR1
SCHEMBL8717852 0.61 TACR1 (0.46) TACR1
SCHEMBL9966004 0.61 MGLL (0.42) TACR1
SCHEMBL16182215 0.60 TACR1 (0.41) TACR1OPRD1
SCHEMBL10607282 0.60 OPRM1 (0.61) OPRM1OPRD1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880529-A1 SPIRO-KETAL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 1998-12-02 EP claimed
WO-1997030056-A1 SPIRO-KETAL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 1997-08-21 WO claimed