SCHEMBL8722332

SCHEMBL8722332

Nc1nc(N)c([N+](=O)[O-])c(OCc2ccc3c(c2)OCO3)n1

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MGMT P16455 10/20 0.63
CCNA2 P20248 1/20 0.46
CDK2 P24941 1/20 0.46
CCNA1 P78396 1/20 0.46
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
PDE5A O76074 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3309544 0.77 MGMT (1.00) MGMTCCNA2CDK2CCNA1CYP3A4
SCHEMBL8722340 0.77 RAB9A (0.49) MGMTKMT2AMAPT
SCHEMBL8507246 0.71 MGMT (0.65) MGMTCCNA2CDK2CCNA1KMT2A
SCHEMBL1154297 0.70 DCPS (0.63) KMT2ATDP1L3MBTL1
SCHEMBL9392819 0.70 CYP3A4 (0.56) KMT2ATDP1L3MBTL1CYP3A4MAPT
SCHEMBL18552099 0.69 ALDH1A1 (0.53)
SCHEMBL3584203 0.68 KMT2A (0.49) KMT2ATDP1L3MBTL1CYP3A4MAPT
SCHEMBL1520844 0.67 CYP3A4 (0.60) KMT2ATDP1L3MBTL1CYP3A4MAPT
SCHEMBL27612725 0.67 CD274 (0.46) MAPT
SCHEMBL6937625 0.67 MAPT (0.46) KMT2ATDP1CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874848-A1 PYRIMIDINE DERIVATIVES AND GUANINE DERIVATIVES, AND THEIR USE IN TREATING TUMOUR CELLS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1998-11-04 EP disclosed
WO-1997020843-A1 PYRIMIDINE DERIVATIVES AND GUANINE DERIVATIVES, AND THEIR USE IN TREATING TUMOUR CELLS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1997-06-12 WO disclosed