SCHEMBL8722720

SCHEMBL8722720

NC(=O)c1ccnc(Oc2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.49
ICAM1 P05362 1/20 0.46
SELE P16581 1/20 0.46
CHEK2 O96017 1/20 0.45
KDM4E B2RXH2 1/20 0.45
KMT2A Q03164 2/20 0.45
USP2 O75604 1/20 0.45
SCN9A Q15858 5/20 0.44
P2RY1 P47900 2/20 0.43
EGFR P00533 1/20 0.43
BTK Q06187 1/20 0.43
ALDH1A1 P00352 2/20 0.43
POLB P06746 2/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAOB P27338 1/20 0.43
F10 P00742 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8721822 0.89 MAPT (0.50) MAPTKDM4EKMT2AP2RY1ALDH1A1
SCHEMBL8722722 0.82 NR3C2 (0.54) MAPTKDM4EP2RY1EGFRALDH1A1
SCHEMBL8569584 0.81 MAPT (0.73) MAPTICAM1SELECHEK2KDM4E
SCHEMBL8721823 0.80 P2RY1 (0.57) MAPTKDM4EKMT2AP2RY1EGFR
SCHEMBL8721009 0.78 MAPT (0.55) MAPTICAM1SELECHEK2KDM4E
SCHEMBL13728192 0.75 KMO (0.52) KDM4ESCN9AALDH1A1
SCHEMBL3844011 0.75 MAPT (0.58) MAPTICAM1SELECHEK2KDM4E
SCHEMBL9233259 0.75 MAPT (0.49) MAPTICAM1SELECHEK2KDM4E
SCHEMBL17242347 0.74 SCN9A (0.44) KDM4ESCN9AF10
SCHEMBL8724391 0.74 CTSS (0.49) MAPTKDM4EKMT2AP2RY1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5759956-A PYRAZINE CARBOXAMIDE DERIVATIVES AMERICAN CYANAMID COMPANY (US) 1998-06-02 US disclosed
EP-0700391-A1 HERBICIDAL COMPOUNDS SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1996-03-13 EP disclosed
WO-1994027974-A1 HERBICIDAL COMPOUNDS SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ B.V. (NL) 1994-12-08 WO disclosed