SCHEMBL8722810

SCHEMBL8722810

CC(C)(C)OC(=O)CC[C@H](NC(=O)c1ccc(N(CCOS(C)(=O)=O)CCOS(C)(=O)=O)c(F)c1)C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TYMS P04818 7/20 0.36
MAPK14 Q16539 1/20 0.34
KDR P35968 1/20 0.34
P2RY12 Q9H244 2/20 0.33
PTPRC P08575 2/20 0.33
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8725881 0.87 TYMS (0.45) TYMSMAPK14KDRP2RY12TAS1R3
SCHEMBL8722803 0.87 TYMS (0.38) TYMSMAPK14KDRP2RY12TAS1R3
SCHEMBL9751797 0.86 P2RY12 (0.38) P2RY12
SCHEMBL8723947 0.85 TYMS (0.35) TYMSP2RY12
SCHEMBL2638361 0.82 TYMS (0.51) TYMSMAPK14
SCHEMBL8726314 0.80 CA2 (0.49) TYMS
SCHEMBL2638442 0.78 TYMS (0.48) TYMS
SCHEMBL6886320 0.77 HDAC1 (0.44) MAPK14KDRPTPRCTAS1R3TAS1R1
SCHEMBL6886329 0.77 HDAC1 (0.44) MAPK14KDRPTPRCTAS1R3TAS1R1
SCHEMBL8726218 0.77 CA2 (0.48) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696270-B1 4-AMINO-FLUOROBENZAMIDES AND THEIR USE AS CYTOTOXIC PRODRUGS CANCER RES CAMPAIGN TECH (GB) 1998-11-04 EP disclosed