SCHEMBL872299

SCHEMBL872299

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)[C@@H]3CCCN3Cc3ccccc3)cc2)cc1)[C@@H]1CCCN1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
PFKFB2 O60825 2/20 0.45
PFKFB1 P16118 2/20 0.45
PFKFB3 Q16875 2/20 0.45
NPSR1 Q6W5P4 1/20 0.44
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
HSD17B10 Q99714 1/20 0.42
KDM1A O60341 1/20 0.41
RCOR1 Q9UKL0 1/20 0.41
GAA P10253 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MEN1 O00255 1/20 0.40
PABPC1 P11940 1/20 0.40
USP2 O75604 1/20 0.40
FKBP1A P62942 1/20 0.40
DPP4 P27487 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845346 0.91 ALDH1A1 (0.53) ALDH1A1NPSR1KMT2AKDM4ELMNA
SCHEMBL13272391 0.91 ALDH1A1 (0.53) ALDH1A1NPSR1KMT2AKDM4ELMNA
SCHEMBL845110 0.86 ALDH1A1 (0.48) ALDH1A1PFKFB2PFKFB1PFKFB3KMT2A
SCHEMBL845507 0.82 F2 (0.50) ALDH1A1PFKFB2PFKFB1PFKFB3KMT2A
SCHEMBL871691 0.81 ALDH1A1 (0.44) ALDH1A1PFKFB2PFKFB1PFKFB3KMT2A
SCHEMBL10119320 0.81 ALDH1A1 (0.43) ALDH1A1PFKFB2PFKFB1PFKFB3KMT2A
SCHEMBL874311 0.80 ALDH1A1 (0.47) ALDH1A1PFKFB2PFKFB1PFKFB3KMT2A
SCHEMBL873465 0.79 KDM4E (0.47) ALDH1A1PFKFB2PFKFB1PFKFB3NPSR1
SCHEMBL10119592 0.79 F2 (0.43) ALDH1A1KMT2ALMNACYP2C9MEN1
SCHEMBL872886 0.78 KDM4E (0.52) ALDH1A1PFKFB2PFKFB1PFKFB3NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed