SCHEMBL845507

SCHEMBL845507

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)C3Cc4ccccc43)cc2)cc1)[C@@H]1CCCN1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 3/20 0.50
ALDH1A1 P00352 3/20 0.40
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HDAC8 Q9BY41 2/20 0.39
PABPC1 P11940 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
DPP4 P27487 4/20 0.38
SCN3A Q9NY46 2/20 0.38
SCN9A Q15858 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845003 0.91 F2 (0.58) F2ALDH1A1CYP2C9CYP2C19PABPC1
SCHEMBL872299 0.82 ALDH1A1 (0.45) ALDH1A1CYP2C9CYP2C19PABPC1DPP4
SCHEMBL845110 0.81 ALDH1A1 (0.48) ALDH1A1CYP2C9CYP2C19PFKFB2PFKFB1
SCHEMBL10119592 0.79 F2 (0.43) F2ALDH1A1CYP2C9SCN3ASCN9A
SCHEMBL872886 0.79 KDM4E (0.52) ALDH1A1PABPC1MAPK1HTTPFKFB2
SCHEMBL10119315 0.79 MAPT (0.40) ALDH1A1CYP2C9CYP2C19SCN3ASCN9A
SCHEMBL874056 0.79 TRPV1 (0.42) ALDH1A1CYP2C9CYP2C19MAPK1HTT
SCHEMBL844873 0.78 NPC1 (0.63) ALDH1A1HDAC8PABPC1DPP4SCN3A
SCHEMBL10119687 0.78 CYP2C9 (0.44) ALDH1A1CYP2C9CYP2C19HDAC8PABPC1
SCHEMBL10119642 0.77 HDAC3 (0.40) ALDH1A1CYP2C9CYP2C19HDAC8HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed