SCHEMBL8723261

SCHEMBL8723261

O=c1[nH]ncn1-c1ccc(N2CCN(c3ccc(OCC(F)(F)C(F)F)cc3)CC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.41
HTT P42858 4/20 0.41
GPR119 Q8TDV5 1/20 0.40
CACNA1G O43497 2/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ALDH1A1 P00352 3/20 0.38
MMP13 P45452 1/20 0.37
MMP14 P50281 1/20 0.37
MAPT P10636 1/20 0.36
LMNA P02545 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ENPP2 Q13822 1/20 0.34
CMA1 P23946 1/20 0.34
KCNH2 Q12809 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6174527 0.93 HTT (0.46) ACACBHTTGPR119KMT2ASMN1; SMN2
SCHEMBL7678488 0.87 HTT (0.41) ACACBHTTGPR119KMT2ASMN1; SMN2
SCHEMBL7686964 0.84 HTT (0.39) ACACBHTTGPR119KMT2ASMN1; SMN2
SCHEMBL9232197 0.83 HTT (0.44) HTTGPR119CACNA1GMMP13MMP14
SCHEMBL8718847 0.82 ACACB (0.41) ACACBHTTCACNA1GKMT2ASMN1; SMN2
SCHEMBL9232299 0.80 HTT (0.54) HTTGPR119CMA1TDP1
SCHEMBL8718743 0.79 USP2 (0.46) HTTGPR119KMT2ASMN1; SMN2MAPT
SCHEMBL8721370 0.78 HTT (0.48) HTTGPR119KMT2AMMP13MMP14
SCHEMBL15912908 0.77 GPR119 (0.44) HTTGPR119KMT2AALDH1A1MAPT
SCHEMBL6647622 0.76 ADRB1 (0.50) ACACBHTTKMT2ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0567982-B1 Azole compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-07-01 EP disclosed
US-5466820-A Fungicides TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-14 US disclosed
US-5371101-A Fungicides TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-12-06 US disclosed
EP-0567982-A1 Azole compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1993-11-03 EP disclosed