SCHEMBL9232197

SCHEMBL9232197

O=c1[nH]ncn1-c1ccc(N2CCN(c3ccc(OC(F)(F)C(F)F)cc3)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.44
GPR119 Q8TDV5 1/20 0.40
POLB P06746 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PPARD Q03181 1/20 0.37
PPARA Q07869 1/20 0.37
MAPT P10636 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
KCNA5 P22460 1/20 0.35
LCAT P04180 2/20 0.34
CACNA1G O43497 1/20 0.34
SCN9A Q15858 1/20 0.34
MAP4K1 Q92918 1/20 0.34
CMA1 P23946 1/20 0.34
AKT1 P31749 1/20 0.33
MMP13 P45452 1/20 0.33
MMP14 P50281 1/20 0.33
KCNH2 Q12809 1/20 0.33
HTR7 P34969 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8718390 0.92 HTT (0.50) HTTGPR119POLBL3MBTL1PPARD
SCHEMBL8723261 0.83 ACACB (0.41) HTTGPR119MAPTTDP1CACNA1G
SCHEMBL8718833 0.80 POLB (0.56) HTTGPR119POLBL3MBTL1PPARD
SCHEMBL3117217 0.79 MAPT (0.52) L3MBTL1MAPTTDP1
SCHEMBL6174527 0.74 HTT (0.46) HTTGPR119POLBL3MBTL1MAPT
SCHEMBL29945199 0.74 GAA (0.48) HTTGPR119MAPTTDP1
SCHEMBL14884466 0.74 GPR119 (0.48) HTTGPR119MAPT
SCHEMBL7190990 0.74 KCNA5 (0.36) PPARDPPARAMAPTKCNA5CACNA1G
SCHEMBL20639686 0.74 GPR119 (0.48) HTTGPR119MAPTMMP13
SCHEMBL3937241 0.74 ADRB1 (0.56) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0659751-A1 Optically active azole derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-06-28 EP disclosed