SCHEMBL8723295

SCHEMBL8723295

COC(=O)c1cccc(CN2CCN(c3cccc(C(F)(F)F)n3)CC2)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.52
DRD2 P14416 3/20 0.49
DRD3 P35462 3/20 0.49
DRD4 P21917 1/20 0.49
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
HTR2B P41595 1/20 0.49
OPRM1 P35372 1/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HSD17B10 Q99714 1/20 0.48
PHGDH O43175 2/20 0.45
GNRHR P30968 1/20 0.45
ACKR3 P25106 5/20 0.44
CHRM3 P20309 1/20 0.44
FAAH O00519 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7109637 0.89 HTR1A (0.52) HTR1ADRD2DRD3DRD4HTR2A
SCHEMBL7184572 0.80 ALDH1A1 (0.62) HTR1ADRD2DRD3OPRM1MEN1
SCHEMBL18998015 0.79 KDM4E (0.63) MEN1KMT2AALDH1A1HSD17B10PHGDH
SCHEMBL7183141 0.79 ALDH1A1 (0.57) HTR1ADRD2DRD3DRD4OPRM1
SCHEMBL6858059 0.79 KDM4E (0.59) HTR1ADRD2DRD3DRD4OPRM1
SCHEMBL6863207 0.79 DRD2 (0.54) HTR1ADRD2DRD3DRD4OPRM1
SCHEMBL6858056 0.78 ALDH1A1 (0.54) MEN1KMT2AALDH1A1SMN1; SMN2FAAH
SCHEMBL27040179 0.77 HTR7 (0.62) DRD4MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL10145077 0.76 ALDH1A1 (0.60) MEN1KMT2AALDH1A1SMN1; SMN2HSD17B10
SCHEMBL31721209 0.76 ALDH1A1 (0.60) MEN1KMT2AALDH1A1SMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998020349-A1 COMPLEX CHEMICAL LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-05-14 WO disclosed