SCHEMBL8724176

SCHEMBL8724176

Cc1ccc(-c2cc(-n3ccnc3)c(-n3ccnc3)s2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
GAA P10253 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ADH5 P11766 4/20 0.37
CYP19A1 P11511 4/20 0.37
CYP11B1 P15538 2/20 0.37
CYP11B2 P19099 2/20 0.37
IDO1 P14902 4/20 0.36
KMT2A Q03164 2/20 0.36
CD38 P28907 1/20 0.36
MEN1 O00255 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PDE3B Q13370 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8722249 0.87 IDO1 (0.39) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8726103 0.85 MEN1 (0.49) CYP1A2CYP3A4GAACYP2D6CYP2C9
SCHEMBL8726099 0.75 PKM (0.41) CYP1A2CYP3A4GAACYP2C9CYP2C19
SCHEMBL8724299 0.71 IDO1 (0.49) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8721485 0.70 NOTUM (0.47) CYP1A2CYP3A4CYP2D6ADH5CYP19A1
SCHEMBL19186987 0.70 KMT2A (0.70) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8720881 0.70 MEN1 (0.47) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL2666052 0.69 CYP19A1 (0.45) CYP1A2CYP3A4GAACYP2D6CYP2C9
SCHEMBL11569176 0.68 IDO1 (0.44) CYP1A2CYP3A4GAACYP2D6CYP2C9
SCHEMBL1885632 0.68 CYP3A4 (0.46) CYP1A2CYP3A4GAACYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998000430-A1 IMIDAZOL DERIVATIVES USEFUL AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-01-08 WO disclosed