SCHEMBL8725201

SCHEMBL8725201

CCOC(=O)c1cnc(NC(=O)/C(=C\C=O)CN)nc1C(F)(F)C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
NFKB1 P19838 7/20 0.46
JUN P05412 6/20 0.46
NFKB2 Q00653 6/20 0.46
RELA Q04206 6/20 0.46
RAB9A P51151 3/20 0.39
NPSR1 Q6W5P4 1/20 0.39
NPC1 O15118 2/20 0.39
MAPT P10636 1/20 0.39
FOS P01100 3/20 0.36
CSNK1D P48730 1/20 0.36
HSP90AA1 P07900 1/20 0.35
DPP4 P27487 2/20 0.35
ALDH1A1 P00352 2/20 0.35
PKM P14618 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ATF1 P18846 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8721324 0.93 KDM4E (0.56) KDM4ENFKB1JUNNFKB2RELA
SCHEMBL8721355 0.91 MAPT (0.41) KDM4ENFKB1JUNNFKB2RELA
SCHEMBL8721300 0.86 RAB9A (0.52) KDM4ENFKB1JUNNFKB2RELA
SCHEMBL8726399 0.84 RAB9A (0.42) KDM4ENFKB1JUNNFKB2RELA
SCHEMBL8889739 0.83 MAPT (0.48) KDM4ENFKB1JUNNFKB2RELA
SCHEMBL8725171 0.83 NFKB1 (0.52) KDM4ENFKB1JUNNFKB2RELA
SCHEMBL8724454 0.82 HSP90AA1 (0.55) KDM4ENFKB1JUNNFKB2RELA
SCHEMBL8891103 0.81 NFKB1 (0.52) KDM4ENFKB1JUNNFKB2RELA
SCHEMBL8721404 0.81 NFKB1 (0.42) KDM4ENFKB1JUNNFKB2RELA
SCHEMBL8395161 0.81 KDM4E (0.56) KDM4ENFKB1JUNNFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998038171-A1 PYRIMIDINE CARBOXYLATES AND RELATED COMPOUNDS AND METHODS FOR TREATING INFLAMMATORY CONDITIONS SIGNAL PHARMACEUTICALS, INC. (US) 1998-09-03 WO claimed
WO-1998038171-A1 PYRIMIDINE CARBOXYLATES AND RELATED COMPOUNDS AND METHODS FOR TREATING INFLAMMATORY CONDITIONS SIGNAL PHARMACEUTICALS, INC. (US) 1998-09-03 WO disclosed
WO-1997009325-A1 PYRIMIDINE CARBOXYLATES AND RELATED COMPOUNDS AND METHODS FOR TREATING INFLAMMATORY CONDITIONS SIGNAL PHARMACEUTICALS, INC. (US) 1997-03-13 WO disclosed