SCHEMBL8891103

SCHEMBL8891103

CC(C)(C)OC(=O)c1cnc(NC(=O)/C(=C\C=O)CN)nc1C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 7/20 0.52
JUN P05412 4/20 0.52
NFKB2 Q00653 4/20 0.52
RELA Q04206 4/20 0.52
KDM4E B2RXH2 1/20 0.40
MAPT P10636 2/20 0.39
GAA P10253 2/20 0.38
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
CNR2 P34972 8/20 0.33
ATF1 P18846 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8889739 0.91 MAPT (0.48) NFKB1JUNNFKB2RELAKDM4E
SCHEMBL8721324 0.88 KDM4E (0.56) NFKB1JUNNFKB2RELAKDM4E
SCHEMBL8888457 0.85 CNR2 (0.39) NFKB1JUNNFKB2RELAKDM4E
SCHEMBL8721355 0.83 MAPT (0.41) NFKB1JUNNFKB2RELAKDM4E
SCHEMBL8725201 0.81 KDM4E (0.47) NFKB1JUNNFKB2RELAKDM4E
SCHEMBL8722111 0.78 NFKB1 (0.60) NFKB1JUNNFKB2RELAKDM4E
SCHEMBL8721300 0.74 RAB9A (0.52) NFKB1JUNNFKB2RELAKDM4E
SCHEMBL8726399 0.72 RAB9A (0.42) NFKB1JUNNFKB2RELAKDM4E
SCHEMBL8725171 0.72 NFKB1 (0.52) NFKB1JUNNFKB2RELAKDM4E
SCHEMBL8724454 0.70 HSP90AA1 (0.55) NFKB1JUNNFKB2RELAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997009325-A1 PYRIMIDINE CARBOXYLATES AND RELATED COMPOUNDS AND METHODS FOR TREATING INFLAMMATORY CONDITIONS SIGNAL PHARMACEUTICALS, INC. (US) 1997-03-13 WO disclosed