SCHEMBL8726720

SCHEMBL8726720

COc1ccc2c(c1OC)C(=Cc1ccccc1)OC2=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.50
KDM4E B2RXH2 6/20 0.50
HPGD P15428 5/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
SMN1; SMN2 Q16637 3/20 0.49
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
POLB P06746 2/20 0.47
MAPT P10636 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C19 P33261 2/20 0.46
STK17B O94768 3/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13239956 0.83 ALDH1A1 (0.58) ALDH1A1KDM4EHPGDL3MBTL1TDP1
SCHEMBL4226377 0.77 RAB9A (0.57) ALDH1A1KDM4EHPGDTDP1SMN1; SMN2
SCHEMBL10618299 0.77 TRPA1 (0.52) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL10618307 0.77 TRPA1 (0.52) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL8724175 0.77 KDM4E (0.60) ALDH1A1KDM4EHPGDL3MBTL1TDP1
SCHEMBL8724172 0.77 KDM4E (0.60) ALDH1A1KDM4EHPGDL3MBTL1TDP1
SCHEMBL7970058 0.72 SMN1; SMN2 (0.49) ALDH1A1KDM4ETDP1SMN1; SMN2NPC1
SCHEMBL7970055 0.72 SMN1; SMN2 (0.49) ALDH1A1KDM4ETDP1SMN1; SMN2NPC1
SCHEMBL30395765 0.71 KDM4E (0.61) ALDH1A1KDM4EHPGDL3MBTL1TDP1
SCHEMBL28996362 0.71 KDM4E (0.61) ALDH1A1KDM4EHPGDL3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883609-A1 SELECTIVE D1 DOPAMINE RECEPTOR AGONISTS AND PARTIAL AGONISTS/ANTAGONISTS Pharmeco Laboratories, Inc. (US) 1998-12-16 EP disclosed
WO-1997030977-A1 SELECTIVE D1 DOPAMINE RECEPTOR AGONISTS AND PARTIAL AGONISTS/ANTAGONISTS PHARM-ECO LABORATORIES, INCORPORATED (US) 1997-08-28 WO disclosed