SCHEMBL8727254

SCHEMBL8727254

CC(C)(C)n1cnc2c(Cl)nc3ccccc3c21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 6/20 0.43
PDE4D Q08499 2/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
HRH2 P25021 1/20 0.39
ADRA1D P25100 1/20 0.39
HTR2A P28223 1/20 0.39
ADORA2A P29274 1/20 0.39
ADRA1A P35348 1/20 0.39
NUDT1 P36639 1/20 0.39
HTR2B P41595 1/20 0.39
KCNH2 Q12809 1/20 0.39
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
ATM Q13315 1/20 0.35
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
METAP1 P53582 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8727241 0.85 TLR7 (0.44) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL8725704 0.82 TLR7 (0.46) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL8723784 0.82 TLR7 (0.62) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL9601821 0.80 IKBKB (0.46) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL8722638 0.78 TLR7 (0.39) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL4758842 0.77 TLR7 (0.42) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL1895460 0.77 TLR7 (0.73) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL10732746 0.77 TLR7 (0.51) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL24499504 0.76 PI4KA (0.39) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL10731424 0.76 FGFR1 (0.46) TLR7PDE4DLMNAPOLBHRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756747-A 1H-imidazo 4,5-c!quinolin-4-amines RIKER LABORATORIES, INC. (US) 1998-05-26 US disclosed
EP-0385630-B1 1H-imidazo(4,5-c)Quinolin-4-amines as antivirals RIKER LABORATORIES INC (US) 1996-11-27 EP disclosed
EP-0389302-B1 Olefinic 1H-imidazo [4,5-c]quinolin-4-amines RIKER LABORATORIES INC (US) 1994-08-31 EP disclosed
US-5037986-A Olefinic 1H-imidazo[4,5-c]quinolin-4-amines MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1991-08-06 US disclosed
EP-0389302-A1 Olefinic 1H-imidazo [4,5-c]quinolin-4-amines RIKER LABORATORIES, INC. (US) 1990-09-26 EP disclosed
EP-0385630-A2 1H-imidazo(4,5-c)Quinolin-4-amines as antivirals RIKER LABORATORIES, INC. (US) 1990-09-05 EP disclosed