SCHEMBL8728949

SCHEMBL8728949

[CH2]CN1CCC(NCC)CC1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.38
ACHE P22303 3/20 0.33
BACE1 P56817 3/20 0.33
CCR5 P51681 1/20 0.33
BCHE P06276 1/20 0.33
CARM1 Q86X55 1/20 0.33
PRMT6 Q96LA8 1/20 0.33
GNAI3 P08754 1/20 0.31
GNAO1 P09471 1/20 0.31
GNAI1 P63096 1/20 0.31
DPP7 Q9UHL4 1/20 0.31
AKT1 P31749 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8728946 0.83 CARM1 (0.37) KCNH2CCR5CARM1PRMT6GNAI3
SCHEMBL2760188 0.82 SMN1; SMN2 (0.42) KCNH2ACHEBACE1CCR5BCHE
SCHEMBL22878502 0.78 PABPC1 (0.46) KCNH2CARM1PRMT6GNAI3GNAO1
SCHEMBL8488055 0.77 KCNH2 (0.40) KCNH2AKT1
SCHEMBL5789303 0.77 CARM1 (0.34) CARM1PRMT6
SCHEMBL12464451 0.77 ACHE (0.44) KCNH2ACHE
SCHEMBL24673647 0.75 ROCK2 (0.39) KCNH2ACHEBACE1CCR5BCHE
SCHEMBL19723131 0.75 KDM1A (0.42) KCNH2CARM1PRMT6GNAI3GNAO1
SCHEMBL27969225 0.75 KCNH2 (0.35) KCNH2ACHEBACE1CCR5BCHE
SCHEMBL4572196 0.75 DPP7 (0.44) KCNH2GNAI3GNAO1GNAI1DPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0624584-B1 Piperazine derivatives useful as calmodulin inhibitors DAIICHI SEIYAKU CO (JP) 1998-08-19 EP disclosed
US-5681954-A HAS CALMODULIN INHIBITORY ACTIVITY; USEFUL IN TREATING DISEASES OF THE CIRCULATORY ORGANS OR IN CEREBRAL REGION DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-10-28 US disclosed
EP-0624584-A1 Piperazine derivatives useful as calmodolin inhibitors DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1994-11-17 EP disclosed