SCHEMBL8729136

SCHEMBL8729136

C[C@@H](Cc1ccccc1CP(=O)(O)COc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HDAC8 Q9BY41 1/20 0.43
CTSS P25774 8/20 0.41
CTSK P43235 8/20 0.41
CTSL P07711 2/20 0.40
CTSB P07858 2/20 0.40
ATM Q13315 1/20 0.39
BCL2 P10415 1/20 0.39
PTPN1 P18031 1/20 0.39
SCN9A Q15858 1/20 0.38
MTNR1A P48039 3/20 0.38
MTNR1B P49286 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8729143 1.00 CYP2C9 (0.44) CYP2C9CYP2C19HDAC8CTSSCTSK
SCHEMBL8729117 0.79 HDAC8 (0.47) HDAC8CTSSCTSKCTSLCTSB
SCHEMBL5586793 0.77 CTSK (0.49) CTSSCTSKCTSLCTSBATM
SCHEMBL8729106 0.77 ADRB3 (0.49) HDAC8CTSSCTSKCTSLCTSB
SCHEMBL8729115 0.77 ADRB3 (0.49) HDAC8CTSSCTSKCTSLCTSB
SCHEMBL8729119 0.75 ACACB (0.49) HDAC8PTPN1
SCHEMBL8732286 0.75 ACACB (0.49) HDAC8PTPN1
SCHEMBL8729003 0.75 ACACB (0.49) HDAC8PTPN1
SCHEMBL507002 0.75 MTNR1A (0.66) CTSSCTSKATMMTNR1AMTNR1B
SCHEMBL507001 0.75 MTNR1A (0.66) CTSSCTSKATMMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726165-A HYPOGLYCEMIC AGENTS; DIETETICS; GASTROINTESTINAL DISORDERS SMITHKLINE BEECHAM P.L.C. (GB) 1998-03-10 US disclosed