SCHEMBL8732121

SCHEMBL8732121

CN(Cc1ccccc1)C(=O)c1ccc(C(=O)c2ccc(CC(=O)O)n2C)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCL8 P10145 1/20 0.61
AKR1B1 P15121 1/20 0.61
PTGS1 P23219 1/20 0.61
PTGS2 P35354 1/20 0.61
GLO1 Q04760 1/20 0.61
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
MLYCD O95822 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
LIMK2 P53671 2/20 0.46
MAOA P21397 1/20 0.46
HPGD P15428 3/20 0.46
ABL1 P00519 1/20 0.46
LCK P06239 1/20 0.46
LIMK1 P53667 1/20 0.46
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
TSHR P16473 1/20 0.44
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8726746 0.86 PTGS2 (0.65) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL8728764 0.83 CXCL8 (0.64) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL8731019 0.82 PTGS2 (0.70) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL8729681 0.82 PTGS2 (0.70) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL8726561 0.82 PTGS2 (0.78) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL2237360 0.82 PTGS2 (0.77) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL8726749 0.80 PTGS2 (0.67) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL8458232 0.79 PTGS1 (0.74) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL14812071 0.78 HDAC1 (0.64) AKR1B1MEN1KMT2AMLYCDHDAC1
SCHEMBL8726505 0.77 CXCL8 (0.62) CXCL8AKR1B1PTGS1PTGS2GLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0783488-A4 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO (JP) 1998-01-07 EP claimed
EP-0783488-A1 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO., LTD. (JP) 1997-07-16 EP claimed
WO-1996010013-A1 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO., LTD. (JP) 1996-04-04 WO claimed