SCHEMBL8726746

SCHEMBL8726746

Cn1c(CC(=O)O)ccc1C(=O)c1ccc(CN(Cc2ccccc2)Cc2ccccc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.65
CXCL8 P10145 1/20 0.65
AKR1B1 P15121 1/20 0.65
PTGS1 P23219 1/20 0.65
GLO1 Q04760 1/20 0.65
HPGD P15428 1/20 0.49
ACHE P22303 8/20 0.42
BCHE P06276 3/20 0.42
HSP90AB1 P08238 1/20 0.40
PTPN1 P18031 1/20 0.40
ABCB11 O95342 1/20 0.39
SRD5A2 P31213 1/20 0.39
NR1H4 Q96RI1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8729681 0.88 PTGS2 (0.70) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL8731019 0.88 PTGS2 (0.70) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL8732121 0.86 CXCL8 (0.61) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL8726561 0.85 PTGS2 (0.78) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL2237360 0.85 PTGS2 (0.77) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL8458232 0.82 PTGS1 (0.74) PTGS2CXCL8AKR1B1PTGS1GLO1
Water SCHEMBL9275860 0.81 PTGS2 (0.72) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL8733588 0.80 CXCL8 (0.62) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL8726505 0.80 CXCL8 (0.62) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL8728778 0.80 CXCL8 (0.52) PTGS2CXCL8AKR1B1PTGS1GLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0783488-A4 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO (JP) 1998-01-07 EP claimed
EP-0783488-A1 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO., LTD. (JP) 1997-07-16 EP claimed
WO-1996010013-A1 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO., LTD. (JP) 1996-04-04 WO claimed