SCHEMBL8733133

SCHEMBL8733133

CCCC(NCC(O)COc1ccc(OCc2ccccc2)c(OCc2ccccc2)c1)(Oc1ccccc1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 5/20 0.47
ADRB2 P07550 1/20 0.45
ADRB1 P08588 1/20 0.45
ADRB3 P13945 1/20 0.45
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
CYP2D6 P10635 2/20 0.42
RAD52 P43351 2/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
CASR P41180 6/20 0.41
KCNH2 Q12809 2/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
C5AR1 P21730 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8728061 0.85 ADRB2 (0.49) ADRB2ADRB1ADRB3ITGB3ITGA2B
SCHEMBL8734022 0.84 CYP2D6 (0.52) ADRB2ADRB1ADRB3ITGB3ITGA2B
SCHEMBL8733140 0.84 KDM4E (0.42) ABCB1KMT2AMEN1KDM4ELMNA
SCHEMBL8733094 0.80 ADRB3 (0.46) ADRB2ADRB1ADRB3CYP2D6RAD52
SCHEMBL9330596 0.76 CYP2D6 (0.60) ADRB2ADRB1ADRB3ITGB3ITGA2B
SCHEMBL23403561 0.75 RAB9A (0.50) ABCB1ADRB2ADRB1ADRB3CYP2D6
SCHEMBL22806689 0.75 ABCB1 (0.52) ABCB1ADRB2ADRB1ADRB3KMT2A
SCHEMBL22806688 0.75 ABCB1 (0.52) ABCB1ADRB2ADRB1ADRB3KMT2A
SCHEMBL21634023 0.74 ADRB2 (0.63) ADRB2ADRB1ADRB3CYP2D6SLC6A2
SCHEMBL29721075 0.74 ADRB2 (0.63) ADRB2ADRB1ADRB3CYP2D6SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726165-A HYPOGLYCEMIC AGENTS; DIETETICS; GASTROINTESTINAL DISORDERS SMITHKLINE BEECHAM P.L.C. (GB) 1998-03-10 US disclosed