SCHEMBL8738529

SCHEMBL8738529

CCCCc1ccnc(-c2cc(CCCC)cc(-c3cc(CCCC)ccn3)n2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
MAPK1 P28482 3/20 0.43
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
SKP2 Q13309 1/20 0.40
TLR8 Q9NR97 1/20 0.39
CTRC Q99895 1/20 0.38
NFKB1 P19838 4/20 0.37
NFKB2 Q00653 3/20 0.37
RELA Q04206 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
L3MBTL1 Q9Y468 3/20 0.37
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.37
CCR1 P32246 1/20 0.36
CCR5 P51681 1/20 0.36
CCR8 P51685 1/20 0.36
PSMB5 P28074 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10020880 0.93 PTGS2 (0.44) NPC1RAB9ASMN1; SMN2L3MBTL1TP53
SCHEMBL2993441 0.93 SKP2 (0.44) NPC1RAB9AMAPK1HPGDHTT
SCHEMBL1146845 0.91 SKP2 (0.43) NPC1RAB9AMAPK1HPGDHTT
SCHEMBL29191290 0.86 SKP2 (0.40) NPC1RAB9AMAPK1HPGDHTT
SCHEMBL12993222 0.85 PTGS2 (0.41) NPC1RAB9ASMN1; SMN2L3MBTL1TP53
SCHEMBL11798255 0.85 TDP1 (0.46) NPC1RAB9AHPGDSMN1; SMN2L3MBTL1
SCHEMBL1446914 0.85 TDP1 (0.46) NPC1RAB9AHPGDSMN1; SMN2L3MBTL1
SCHEMBL913250 0.85 TDP1 (0.46) NPC1RAB9AHPGDSMN1; SMN2L3MBTL1
SCHEMBL7963811 0.85 TDP1 (0.46) NPC1RAB9AHPGDSMN1; SMN2L3MBTL1
SCHEMBL7964430 0.85 TDP1 (0.46) NPC1RAB9AHPGDSMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9708336-B2 Metallo-beta-lactamase inhibitors MERCK SHARP & DOHME CORP. (US) 2017-07-18 US disclosed
WO-2012065981-A1 COMPOUND OR MIXTURE OF PHOTOLUMINESCENT COMPOUNDS ENI S.P.A. (IT) 2012-05-24 WO disclosed