SCHEMBL874280

SCHEMBL874280

O=C(Nc1ccc(-c2ccc(C(=O)NCCC3CCCCC3)c(Nc3ccccc3)n2)cc1)c1cc2cccnc2s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
GAA P10253 1/20 0.38
CHRNA7 P36544 2/20 0.36
NAMPT P43490 1/20 0.36
RAB9A P51151 2/20 0.36
KIT P10721 2/20 0.36
MAPK14 Q16539 2/20 0.36
NPC1 O15118 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ADORA2A P29274 1/20 0.35
CAMKK1 Q8N5S9 1/20 0.35
CAMKK2 Q96RR4 1/20 0.35
SYK P43405 1/20 0.35
MAPK1 P28482 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL873721 0.90 BCHE (0.39) BCHEACHECHRNA7NAMPTRAB9A
SCHEMBL873820 0.87 ATR (0.46) MEN1KMT2ACHRNA7NAMPTNPSR1
SCHEMBL873584 0.85 KMT2A (0.40) MEN1KMT2AALDH1A1MAPTGAA
SCHEMBL874281 0.83 RAB9A (0.40) MEN1KMT2AALDH1A1MAPTGAA
SCHEMBL874835 0.82 MEN1 (0.43) MEN1KMT2AALDH1A1MAPTGAA
SCHEMBL875500 0.79 ATR (0.41) CHRNA7NAMPTSYKNPSR1
SCHEMBL873865 0.79 NAMPT (0.42) BCHEACHEALDH1A1GAACHRNA7
SCHEMBL873821 0.78 NAMPT (0.39) MEN1KMT2AALDH1A1MAPTGAA
SCHEMBL874291 0.78 CHRNA7 (0.39) BCHEACHEKMT2AMAPTCHRNA7
SCHEMBL874482 0.77 CHRM4 (0.42) BCHEACHEMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed