SCHEMBL874409

SCHEMBL874409

CCCCc1nc(-c2ccc(N)cc2)sc1C(=O)NCCN1CCOCC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 4/20 0.55
ALDH1A1 P00352 6/20 0.50
HSD17B10 Q99714 5/20 0.50
HPGD P15428 5/20 0.50
KDM4E B2RXH2 4/20 0.50
CASP1 P29466 4/20 0.50
CASP7 P55210 4/20 0.50
GAA P10253 3/20 0.50
TSHR P16473 3/20 0.50
GLA P06280 3/20 0.50
USP2 O75604 3/20 0.50
NPSR1 Q6W5P4 3/20 0.50
MAPT P10636 4/20 0.49
HTT P42858 3/20 0.49
L3MBTL1 Q9Y468 3/20 0.49
LMNA P02545 3/20 0.49
TP53 P04637 2/20 0.49
ALOX15 P16050 2/20 0.49
RECQL P46063 1/20 0.49
CYP1A2 P05177 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874805 0.81 MAPT (0.43) ALDH1A1HSD17B10HPGDKDM4ECASP1
SCHEMBL882713 0.80 CYP3A4 (0.44) CD274ALDH1A1HSD17B10HPGDKDM4E
SCHEMBL874282 0.79 SMN1; SMN2 (0.47) ALDH1A1KDM4EGAAMAPTHTT
SCHEMBL874795 0.75 NAMPT (0.47)
SCHEMBL12336010 0.74 CD274 (0.60) CD274HPGDHTTLMNACYP1A2
SCHEMBL10069158 0.72 CD274 (0.41) CD274ALDH1A1HSD17B10HPGDTSHR
SCHEMBL873629 0.71 NAMPT (0.42)
SCHEMBL3543817 0.71 CD274 (0.92) CD274ALDH1A1HPGDKDM4ETSHR
SCHEMBL15626281 0.69 LMNA (0.55) CD274HPGDLMNAKMT2A
SCHEMBL298546 0.69 MAPK1 (0.56) ALDH1A1HSD17B10HPGDKDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed