SCHEMBL8744759

SCHEMBL8744759

CCOC(=O)[C@@H](NC(=O)Cc1c(C)cc(C)cc1C)[C@@H](C)CC

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.42
GFER P55789 1/20 0.42
LMNA P02545 1/20 0.39
ALDH1A1 P00352 4/20 0.39
TYR P14679 1/20 0.39
ELANE P08246 1/20 0.38
POLB P06746 2/20 0.38
PSMB5 P28074 1/20 0.38
MAPT P10636 1/20 0.38
PYGL P06737 1/20 0.37
CYP2C9 P11712 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
NLRP3 Q96P20 1/20 0.37
HTT P42858 1/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9594066 1.00 KMT2A (0.42) KMT2AGFERLMNAALDH1A1TYR
SCHEMBL9595171 0.90 ALDH1A1 (0.42) KMT2AGFERLMNAALDH1A1PSMB5
SCHEMBL8744786 0.90 ALDH1A1 (0.42) KMT2AGFERLMNAALDH1A1PSMB5
SCHEMBL8744770 0.86 PYGL (0.38) KMT2AGFERLMNAALDH1A1PSMB5
SCHEMBL9596067 0.86 PYGL (0.38) KMT2AGFERLMNAALDH1A1PSMB5
SCHEMBL8744757 0.86 KMT2A (0.54) KMT2AGFERALDH1A1PYGLCYP2C9
SCHEMBL8744747 0.86 KMT2A (0.54) KMT2AGFERALDH1A1PYGLCYP2C9
SCHEMBL9595368 0.84 LMNA (0.41) LMNAPSMB5NLRP3
SCHEMBL8744813 0.84 LMNA (0.41) LMNAPSMB5NLRP3
SCHEMBL7964632 0.84 ALDH1A1 (0.50) KMT2AGFERLMNAALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456063-B1 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1997-01-22 EP disclosed
US-5258527-A Insecticidal, acaricidal and herbicidal 1-H-3-aryl-pyrrolidine-2,4-dione derivatives BAYER AKTIENGESELLSCHAFT (DE) 1993-11-02 US disclosed
EP-0456063-A2 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1991-11-13 EP disclosed