SCHEMBL8744800

SCHEMBL8744800

C[C@H](NC(=O)Cc1c(Cl)cccc1Cl)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.53
KMT2A Q03164 1/20 0.51
SLC22A12 Q96S37 1/20 0.51
ALDH1A1 P00352 3/20 0.49
HPGD P15428 2/20 0.49
POLB P06746 1/20 0.49
HSD17B10 Q99714 1/20 0.48
RECQL P46063 1/20 0.48
SMN1; SMN2 Q16637 4/20 0.46
KDM4E B2RXH2 1/20 0.46
SHMT1 P34896 3/20 0.45
SHMT2 P34897 3/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
SIGMAR1 Q99720 1/20 0.43
PSMB5 P28074 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8744794 1.00 AKR1B1 (0.53) AKR1B1KMT2ASLC22A12ALDH1A1HPGD
SCHEMBL4431531 0.87 SHMT2 (0.51) KMT2ASLC22A12ALDH1A1HPGDPOLB
SCHEMBL4431529 0.87 SHMT2 (0.51) KMT2ASLC22A12ALDH1A1HPGDPOLB
SCHEMBL8744816 0.84 SDCBP (0.51) AKR1B1KMT2ASLC22A12ALDH1A1HPGD
SCHEMBL8744811 0.84 SDCBP (0.51) AKR1B1KMT2ASLC22A12ALDH1A1HPGD
SCHEMBL9594560 0.82 KMT2A (0.47) AKR1B1KMT2ASLC22A12ALDH1A1HPGD
SCHEMBL8744777 0.82 KMT2A (0.47) AKR1B1KMT2ASLC22A12ALDH1A1HPGD
SCHEMBL8744785 0.82 GRN (0.56) AKR1B1KMT2ASLC22A12ALDH1A1
SCHEMBL8744789 0.82 GRN (0.56) AKR1B1KMT2ASLC22A12ALDH1A1
SCHEMBL8744730 0.81 PYGL (0.47) AKR1B1KMT2ASLC22A12ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456063-B1 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1997-01-22 EP disclosed
US-5258527-A Insecticidal, acaricidal and herbicidal 1-H-3-aryl-pyrrolidine-2,4-dione derivatives BAYER AKTIENGESELLSCHAFT (DE) 1993-11-02 US disclosed
EP-0456063-A2 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1991-11-13 EP disclosed