SCHEMBL8744968

SCHEMBL8744968

COC(=O)Cc1ccc(CN2CCN(C(c3ccccc3)c3ccc(Cl)cc3)CC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 5/20 0.64
KCNH2 Q12809 4/20 0.64
ADORA3 P0DMS8 2/20 0.64
CNR1 P21554 2/20 0.64
OPRK1 P41145 2/20 0.64
GHSR Q92847 2/20 0.64
LMNA P02545 2/20 0.64
NR1I2 O75469 1/20 0.64
PDE4D Q08499 1/20 0.64
ATM Q13315 2/20 0.60
CYP3A4 P08684 2/20 0.59
USP2 O75604 2/20 0.59
SLC6A2 P23975 2/20 0.59
HRH2 P25021 2/20 0.59
HTR2A P28223 2/20 0.59
SLC6A4 P31645 2/20 0.59
DRD3 P35462 2/20 0.59
HTR2B P41595 2/20 0.59
SLC6A3 Q01959 2/20 0.59
CYP1A2 P05177 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8690003 0.94 ATM (0.67) HRH1KCNH2ADORA3CNR1OPRK1
SCHEMBL8744969 0.87 ATM (0.67) HRH1KCNH2ADORA3CNR1OPRK1
SCHEMBL12464946 0.84 KCNH2 (0.80) HRH1KCNH2ADORA3CNR1OPRK1
SCHEMBL8744992 0.83 ATM (0.53) HRH1KCNH2ADORA3CNR1OPRK1
SCHEMBL1569388 0.82 KCNH2 (0.70) HRH1KCNH2ADORA3CNR1OPRK1
SCHEMBL588111 0.82 KCNH2 (0.78) HRH1KCNH2ADORA3CNR1OPRK1
SCHEMBL588110 0.82 KCNH2 (0.78) HRH1KCNH2ADORA3CNR1OPRK1
SCHEMBL3611802 0.82 KCNH2 (0.78) HRH1KCNH2ADORA3CNR1OPRK1
SCHEMBL9720751 0.81 KCNH2 (0.71) HRH1KCNH2ADORA3CNR1OPRK1
SCHEMBL8691241 0.81 ATM (0.76) HRH1KCNH2ADORA3CNR1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0753515-A2 Benzylpiperazine derivatives as antiallergic and anti-inflammatory agents Senju Pharmaceutical Co., Ltd. (JP) 1997-01-15 EP claimed
EP-0753515-A2 Benzylpiperazine derivatives as antiallergic and anti-inflammatory agents Senju Pharmaceutical Co., Ltd. (JP) 1997-01-15 EP disclosed