SCHEMBL8744969

SCHEMBL8744969

O=C(O)Cc1ccc(CN2CCN(C(c3ccccc3)c3ccc(Cl)cc3)CC2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.67
HRH1 P35367 5/20 0.67
KCNH2 Q12809 4/20 0.67
ADORA3 P0DMS8 2/20 0.67
CNR1 P21554 2/20 0.67
OPRK1 P41145 2/20 0.67
GHSR Q92847 2/20 0.67
LMNA P02545 2/20 0.67
NR1I2 O75469 1/20 0.67
PDE4D Q08499 1/20 0.67
KDM4E B2RXH2 1/20 0.65
ALDH1A1 P00352 1/20 0.65
MAPT P10636 1/20 0.65
HTT P42858 1/20 0.65
NPSR1 Q6W5P4 1/20 0.65
MEN1 O00255 2/20 0.64
KMT2A Q03164 2/20 0.64
SLC6A9 P48067 1/20 0.64
USP2 O75604 2/20 0.62
CYP3A4 P08684 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8691241 0.94 ATM (0.76) ATMHRH1KCNH2ADORA3CNR1
SCHEMBL12464946 0.89 KCNH2 (0.80) ATMHRH1KCNH2ADORA3CNR1
SCHEMBL8744968 0.87 HRH1 (0.64) ATMHRH1KCNH2ADORA3CNR1
SCHEMBL588111 0.87 KCNH2 (0.78) ATMHRH1KCNH2ADORA3CNR1
SCHEMBL588110 0.87 KCNH2 (0.78) ATMHRH1KCNH2ADORA3CNR1
SCHEMBL3611802 0.87 KCNH2 (0.78) ATMHRH1KCNH2ADORA3CNR1
SCHEMBL9720751 0.86 KCNH2 (0.71) ATMHRH1KCNH2ADORA3CNR1
Hydrochloric Acid SCHEMBL587709 0.85 LMNA (0.79) ATMHRH1KCNH2ADORA3CNR1
Hydrochloric Acid SCHEMBL588103 0.85 LMNA (0.79) ATMHRH1KCNH2ADORA3CNR1
Hydrochloric Acid SCHEMBL588128 0.85 LMNA (0.79) ATMHRH1KCNH2ADORA3CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0753515-A2 Benzylpiperazine derivatives as antiallergic and anti-inflammatory agents Senju Pharmaceutical Co., Ltd. (JP) 1997-01-15 EP claimed
EP-0753515-A2 Benzylpiperazine derivatives as antiallergic and anti-inflammatory agents Senju Pharmaceutical Co., Ltd. (JP) 1997-01-15 EP disclosed